Evolving paradigms in targeting FLT3 for acute myeloid leukemia therapy
  • Thapa, Rajan
  • Shrestha, Jesus
  • Paudel, Keshav Raj
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초록

FLT3 mutations drive acute myeloid leukemia (AML) progression through aberrant signaling, making FLT3 inhibition a key therapeutic strategy. Current inhibitors show efficacy, yet resistance and toxicity remain challenges. Emerging approaches, including selective inhibitors, proteolysis-targeting chimeras, and protein degraders, offer enhanced potency, sustained suppression, and combinatorial potential, representing a precision-based advancement in AML treatment.

키워드

acute myeloid leukemiaantibody-drug conjugatesdrug resistanceFLT3 inhibitors
제목
Evolving paradigms in targeting FLT3 for acute myeloid leukemia therapy
저자
Thapa, RajanShrestha, JesusPaudel, Keshav Raj
DOI
10.1016/j.tips.2026.01.009
발행일
2026-03
유형
Editorial Material
저널명
Trends in Pharmacological Sciences
47
3
페이지
244 ~ 247